<SUBMISSION>
<SECRELEASE-DATETIME> 20170315-163026 ⇐ Metadata from SEC Info (ET)
<SECWEBSITE-DATETIME> 20170315-163026 ⇐ Metadata from SEC Info (ET)
<ACCEPTANCE-DATETIME> 20170315-151952 ⇐ Filing accepted by SEC (ET)
<ACCESSION-NUMBER> 0000799698-17-000012
<TYPE> 10-K
<PUBLIC-DOCUMENT-COUNT> 93
<PERIOD> 20161231
<FILING-DATE> 20170315
<DATE-OF-FILING-DATE-CHANGE> 20170315
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<FILER>
<COMPANY-DATA>
<CONFORMED-NAME> CYTRX CORP
<CIK> 0000799698
<ASSIGNED-SIC> 2836
<IRS-NUMBER> 581642750 ⇒ 58-1642750 or 581-64-2750
<STATE-OF-INCORPORATION> DE
<FISCAL-YEAR-END> 1231
</COMPANY-DATA>
<FILING-VALUES>
<FORM-TYPE> 10-K
<ACT> 34
<FILE-NUMBER> 000-15327
<FILM-NUMBER> 17691050
</FILING-VALUES>
<BUSINESS-ADDRESS>
<STREET1> 11726 SAN VICENTE BOULEVARD
<STREET2> SUITE 650
<CITY> LOS ANGELES
<STATE> CA
<ZIP> 90049
<PHONE> 310-826-5648
</BUSINESS-ADDRESS>
<MAIL-ADDRESS>
<STREET1> 11726 SAN VICENTE BOULEVARD
<STREET2> SUITE 650
<CITY> LOS ANGELES
<STATE> CA
<ZIP> 90049
</MAIL-ADDRESS>
</FILER>
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<DOCUMENT>
<TYPE> 10-K
<SEQUENCE> 1
<FILENAME> 2016_form10-k.htm
<DESCRIPTION> ANNUAL REPORT ON FORM 10-K FOR YEAR ENDING DEC. 31, 2016
<TEXT>
<html>
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<DOCUMENT>
<TYPE> EX-4.6
<SEQUENCE> 2
<FILENAME> exh_4-6.htm
<DESCRIPTION> FORM OF WARRANT DATED JULY 20, 2016
<TEXT>
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<DOCUMENT>
<TYPE> EX-4.7
<SEQUENCE> 3
<FILENAME> exh_4-7.htm
<DESCRIPTION> CONTINGENT COMMON STOCK PURCHASE WARRANT
<TEXT>
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<DOCUMENT>
<TYPE> EX-4.8
<SEQUENCE> 4
<FILENAME> exh_4-8.htm
<DESCRIPTION> EMMANUEL WARRANT ISSUED ON NOVEMBER 10, 2013
<TEXT>
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<DOCUMENT>
<TYPE> EX-4.9
<SEQUENCE> 5
<FILENAME> exh_4-9.htm
<DESCRIPTION> EMMANUEL WARRANT
<TEXT>
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</TEXT>
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<DOCUMENT>
<TYPE> EX-10.26
<SEQUENCE> 6
<FILENAME> exh_10-26.htm
<DESCRIPTION> 2017 EMPLOYMENT AGREEMENT - DANIEL LEVITT, M.D., PH.D.
<TEXT>
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<DOCUMENT>
<TYPE> EX-10.29
<SEQUENCE> 7
<FILENAME> exh_10-29.htm
<DESCRIPTION> 2017 EMPLOYMENT AGREEMENT - SCOTT WIELAND
<TEXT>
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<DOCUMENT>
<TYPE> EX-10.30
<SEQUENCE> 8
<FILENAME> exh_10-30.htm
<DESCRIPTION> 2017 EMPLOYMENT AGREEMENT - JOHN CALOZ
<TEXT>
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<DOCUMENT>
<TYPE> EX-10.31
<SEQUENCE> 9
<FILENAME> exh_10-31.htm
<DESCRIPTION> 2017 EMPLOYMENT AGREEMENT - OLIVIA WARE
<TEXT>
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<DOCUMENT>
<TYPE> EX-10.38
<SEQUENCE> 10
<FILENAME> exh_10-38.htm
<DESCRIPTION> 2017 AMENDMENT TO EMPLOYMENT AGREEMENT - STEVEN A. KRIEGSMAN
<TEXT>
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<DOCUMENT>
<TYPE> EX-10.39
<SEQUENCE> 11
<FILENAME> exh_10-39.htm
<DESCRIPTION> RESTRICTED STOCK PURCHASE AGREEMENT DATED JANUARY 11, 2017
<TEXT>
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<DOCUMENT>
<TYPE> EX-23.1
<SEQUENCE> 12
<FILENAME> exh_23-1.htm
<DESCRIPTION> CONSENT OF INDEPENDENT ACCOUNTING FIRM
<TEXT>
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<DOCUMENT>
<TYPE> EX-31.1
<SEQUENCE> 13
<FILENAME> exh_31-1.htm
<DESCRIPTION> CERTIFICATION OF CHIEF EXECUTIVE OFFICER
<TEXT>
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<DOCUMENT>
<TYPE> EX-31.2
<SEQUENCE> 14
<FILENAME> exh_31-2.htm
<DESCRIPTION> CERTIFICATION OF CHIEF FINANCIAL OFFICER
<TEXT>
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<DOCUMENT>
<TYPE> EX-32.1
<SEQUENCE> 15
<FILENAME> exh_32-1.htm
<DESCRIPTION> CERTIFICATION OF CHIEF EXECUTIVE OFFICER (SEC. 1350)
<TEXT>
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<DOCUMENT>
<TYPE> EX-32.2
<SEQUENCE> 16
<FILENAME> exh_32-2.htm
<DESCRIPTION> CERTIFICATION OF CHIEF FINANCIAL OFFICER (SEC. 1350)
<TEXT>
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<DOCUMENT>
<TYPE> EX-101.LAB
<SEQUENCE> 17
<FILENAME> cytr-20161231_lab.xml
<DESCRIPTION> XBRL TAXONOMY EXTENSION LABEL LINKBASE
<TEXT>
<XBRL>
<?xml version="1.0" encoding="us-ascii"?>
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<TYPE> EX-101.INS
<SEQUENCE> 18
<FILENAME> cytr-20161231.xml
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<TYPE> EX-101.SCH
<SEQUENCE> 19
<FILENAME> cytr-20161231.xsd
<DESCRIPTION> XBRL TAXONOMY EXTENSION SCHEMA
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<TYPE> EX-101.CAL
<SEQUENCE> 20
<FILENAME> cytr-20161231_cal.xml
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<SEQUENCE> 21
<FILENAME> cytr-20161231_def.xml
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<TYPE> EX-101.PRE
<SEQUENCE> 22
<FILENAME> cytr-20161231_pre.xml
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<FILENAME> R12.htm
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<FILENAME> R13.htm
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<FILENAME> R14.htm
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<TEXT>
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<FILENAME> R15.htm
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<TEXT>
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<FILENAME> R16.htm
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<TEXT>
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<FILENAME> R17.htm
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<TEXT>
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<FILENAME> R18.htm
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<TEXT>
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<FILENAME> R19.htm
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<TEXT>
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<FILENAME> R20.htm
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<FILENAME> R21.htm
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<FILENAME> R27.htm
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<FILENAME> R30.htm
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<FILENAME> R31.htm
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<TEXT>
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<FILENAME> R33.htm
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<FILENAME> R34.htm
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<FILENAME> R37.htm
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<DESCRIPTION> IDEA: XBRL DOCUMENT
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<TYPE> XML
<SEQUENCE> 79 ⇐ Document/Exhibit 73
<FILENAME> R51.htm
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<SEQUENCE> 80 ⇐ Document/Exhibit 74
<FILENAME> R52.htm
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<SEQUENCE> 81 ⇐ Document/Exhibit 75
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<SEQUENCE> 82 ⇐ Document/Exhibit 76
<FILENAME> R54.htm
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<SEQUENCE> 83 ⇐ Document/Exhibit 77
<FILENAME> R55.htm
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<SEQUENCE> 84 ⇐ Document/Exhibit 78
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<SEQUENCE> 85 ⇐ Document/Exhibit 79
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<SEQUENCE> 86 ⇐ Document/Exhibit 80
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<SEQUENCE> 87 ⇐ Document/Exhibit 81
<FILENAME> R59.htm
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<SEQUENCE> 88 ⇐ Document/Exhibit 82
<FILENAME> R60.htm
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<SEQUENCE> 89 ⇐ Document/Exhibit 83
<FILENAME> Financial_Report.xlsx
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<TYPE> XML
<SEQUENCE> 90 ⇐ Not a Document/Exhibit
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<SEQUENCE> 91 ⇐ Not a Document/Exhibit
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<TYPE> XML
<SEQUENCE> 93 ⇒ 92 ⇐ Document/Exhibit 84
<FILENAME> FilingSummary.xml
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<SEQUENCE> 95 ⇒ 93 ⇐ Document/Exhibit 85
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<DESCRIPTION> IDEA: XBRL DOCUMENT
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